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Eticlopride (hydrochloride)|29112-10 mg|CAS:97612-24-3
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Eticlopride (hydrochloride)|29112-10 mg|CAS:97612-24-3

29112-10 mg
Eticlopride (hydrochloride)
¥ 1795.6
¥ 1795.6
10 mg
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Eticlopride (hydrochloride)介绍:

产品名称:
Eticlopride (hydrochloride)
别名:
(−)-Eticlopride|S-(−)-Eticlopride
产品描述:
A D2 and D3 receptor antagonist (Kis = 0.029 and 0.46 nM in MN9D mouse neuronal cells expressing rat D2 and human D3 receptors, respectively); selective for dopamine D2 and D3 receptors (IC50s = 1 and 113 nM, respectively) over dopamine D1, α2-adrenergic, and β-adrenergic, Histamine H1, and muscarinic receptors (IC50s = 700->100,000 nM), as well as 5-HT1 and 5-HT2 receptors (IC50s = 6,200 and 830, respectively) in radioligand binding assays; binds α1-ARs (IC50 = 110 nM); inhibits 7-OH-DPAT-induced stereotyped behavior in rats at 10 μg/kg; inhibits inhibits ketamine- and cocaine-induced hypermotility in rats at 20 and 50 μg/kg, respectively
保存温度:
-20
运输温度:
-20
预期分子量:
340.9
产品形式:
A crystalline solid
有效期:
1460
纯度:
≥98%
CAS号:
97612-24-3
分子式:
C17H25ClN2O3 • HCl

本公司销售的所有产品仅供实验科研使用,不用于人体及临床诊断。

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