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Phenamil (methanesulfonate)|14308-10 mg|CAS:1161-94-0
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Phenamil (methanesulfonate)|14308-10 mg|CAS:1161-94-0

14308-10 mg
Phenamil (methanesulfonate)
¥ 1273.0
¥ 1273.0
10 mg
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Phenamil (methanesulfonate)介绍:

产品名称:
Phenamil (methanesulfonate)
产品描述:
A TRPP3 inhibitor (IC50 = 140 nM); also inhibits ENaC (IC50 = 400 nM); decreases basal short-circuit currents in human and ovine bronchial epithelial cells (IC50s = 75 and 116 nM, respectively); inhibits potassium chloride-induced contractions in isolated rat endothelium-denuded aortic rings (EC50 = 6.76 µM) and increases contractile force in isolated rat right ventricular papillary muscles (EC50 = 16.98 µM); reduces pulmonary artery medial wall thickness and decreases right ventricular peak pressure in a rat model of chronic hypoxia-induced pulmonary hypertension at 15 and 30 mg/kg per day
保存温度:
-20
运输温度:
-20
预期分子量:
305.69
产品形式:
A crystalline solid
有效期:
1460
纯度:
≥98%
CAS号:
1161-94-0
分子式:
C12H12ClN7O • CH3SO3H

本公司销售的所有产品仅供实验科研使用,不用于人体及临床诊断。

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